Product Description
CAYMAN CHEMICAL 19375-25 - LENVATINIB - LENVATINIB IS A POTENT INHIBITOR OF VEGF-R2 AND VEGF-R3 KINASE ACTIVITIES WITH IC50 VALUES OF 4.0 AND 5.2 NM, RESPECTIVELY.. IT IS SLIGHTLY LESS POTENT AGAINST THE RELATED RECEPTOR KINASES VEGF-R1, FGF-R1, PGDFR3? AND KIT (IC50 VALUES OF 22, 46, 39, AND 100 NM, RESPECTIVELY). IT IS ORALLY ACTIVE, INHIBITING H136 CELL TUMOR GROWTH IN MICE AT 30 MG/KG. - EQUAL TO C814C18-EA
MANUFACTURER:
CAYMAN CHEMICAL
MANUFACTURER PART NUMBER:
19375-25
UNIT OF MEASURE:
EA
QTY PER UNIT OF MEASURE:
1
COUNTRY OF ORIGIN:
CANADA
ORDER INCREMENT:
1
WEIGHT:
0
CONTRACTOR PART NUMBER:
2800042149